- Oggetto:
- Oggetto:
MOLECULAR MEDICINAL CHEMISTRY
- Oggetto:
Molecular Medicinal Chemistry
- Oggetto:
Academic year 2023/2024
- Course ID
- BIO0186 Pds GEN
- Teacher
- Sonja Visentin
- Degree course
- [0101M22] Molecular Biotechnology
- Year
- 2nd year
- Teaching period
- Second semester
- Type
- Elective
- Credits/Recognition
- 6
- Course disciplinary sector (SSD)
- CHIM/08 - pharmaceutical chemistry
- Delivery
- Formal authority
- Language
- English
- Attendance
- Obligatory
- Type of examination
- Oral
- Type of learning unit
- corso
- Prerequisites
- Basic knowledge of chemistry
- Oggetto:
Sommario del corso
- Oggetto:
Course objectives
What is a drug? This medicinal chemistry course explores how chemists modify a molecule’s structure to design a safe and effective drug.
- Oggetto:
Results of learning outcomes
At the end of the course the student will be able to read critically paper in the field of the drug discovery and have a knowledge of the process that a molecule must do to become a drug
- Oggetto:
Program
Pre-Regulatory Medicine and the Drug Approval Process: Modern drug discovery and approval process for the Intellectual property issues with drugs.
Drug pipeline with some example of drugs that changed the life of patients. Drug screening, Filtering hits to find leads Existing drugs and natural products as leads
Drug Targets: Structure of proteins Enzymes and other targets.
Binding, Structure, and Diversity Intermolecular forces.
Molecular diversity and chemical libraries Combinatorial chemistry
Metabolism: Types of metabolic reactions. How can we use metabolism to obtain safe and effective drugs- Oggetto:
Course delivery
The course will be delivered in blended learning.
Lessons will take place in the classroom or in remote presence according to the guidelines provided by the university.
A student is required to attain at least 75% of the attendance for lectures, tutorials and practical sessions of the course (in classroom or in remote presence).
- Oggetto:
Learning assessment methods
Preparation and discussion of infographics on some topics of the course.
Preparation and discussion of a report on topics related to the program of the course.
Exams will be conducted 'face-to-face' or online according to university guidelines.
- Oggetto:
Support activities
Use of the e-learning platform Moodle
Suggested readings and bibliography
- Oggetto:
The Organic Chemistry of Drug Design and Drug Action
Autore: Richard B. Silverman, Mark W. HollodayEdizione: Third Edition
Casa editrice: Academic Press
ISBN: 9780123820303
Url: https://www.elsevier.com/books/the-organic-chemistry-of-drug-design-and-drug-action/silverman/978-0-12-382030-3The Practice of Medicinal Chemistry
Autore: Camille Wermuth, David Aldous, Pierre Raboisson, Didier RognanEdizione: Fourth Edition
Casa editrice: Academic Press
ISBN: 9780124172050
Url: https://www.elsevier.com/books/the-practice-of-medicinal-chemistry/wermuth/978-0-12-417205-0- Enroll
- Closed
- Enrollment opening date
- 01/03/2020 at 00:00
- Enrollment closing date
- 31/12/2022 at 23:55
- Oggetto:
